Research reference only. Not medical advice. Most compounds are not FDA-approved. Consult a qualified clinician before any human use.

Sexual Function & Libido

Dermorphin

[D-Ala2]-dermorphin

Classification: Opioid peptide (research)

Mechanism: Mu-opioid receptor agonist; BBB-penetrant due to D-amino acids

Benefits: Potent μ-opioid analgesia (30-40x morphine)

Evidence tier: Preclinical + Illicit Use · Availability: Experimental (Illicit)

Primary sources

  1. Schiller PW. Opioid peptide-derived analgesics — discusses dermorphin and DALDA analogues. AAPS J 2005. PMID 16353933
  2. Note: Dermorphin is banned in horse racing and most professional sports as an opioid agonist; human clinical data are limited.

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